InflaRx reports promising data on oral C5aR inhibitor INF904

Published 03/09/2024, 12:50
InflaRx reports promising data on oral C5aR inhibitor INF904

JENA, Germany - InflaRx N.V. (NASDAQ:IFRX), a clinical-stage biopharmaceutical company, has presented preclinical data on its novel oral C5aR inhibitor, INF904, at the European Meeting on Complement in Human Diseases. The data showcased INF904's potential as a strong anti-inflammatory agent with favorable pharmacokinetic properties.

The preclinical studies compared INF904 with avacopan, another C5aR inhibitor. INF904 demonstrated a significant inhibition of C5a-induced neutropenia in a hamster model by 96.5%, a marked improvement over avacopan's 51.1% at the same dose. Additionally, INF904 exhibited 2- to 5-fold higher exposure than avacopan across all tested animal species, suggesting a more favorable pharmacokinetic profile.

INF904 also showed minimal inhibition of the CYP3A4/5 enzymes, which are critical in drug metabolism, including that of glucocorticoids. This characteristic may reduce the likelihood of drug-drug interactions, a significant consideration in developing new medications.

In vitro and in vivo disease models indicated that INF904 reduces neutrophil activation, a key process in inflammation. The inhibitor effectively blocked CD11b upregulation on neutrophils and, after oral dosing, showed significant anti-inflammatory effects in hamster models. These effects included reduced neutrophil influx, decreased plasma levels of CREA and BUN, and histological improvements.

The first-in-human study of INF904 reported that the drug is well-tolerated with no safety concerns at various dosing levels. Pharmacokinetic and pharmacodynamic data from the study support INF904's potential as a leading candidate in the C5aR inhibitor drug class.

Dr. Camilla Chong, Chief Medical Officer of InflaRx, expressed optimism about INF904's differentiating advantages and its alignment with the company's goal to develop first-in-class and best-in-class anti-inflammatory therapies.

InflaRx specializes in anti-inflammatory therapeutics targeting the complement system, with its lead product candidate, vilobelimab, showing clinical activity in multiple studies. The company, founded in 2007, operates from Germany and the United States.

This report is based on a press release statement and does not constitute an endorsement of InflaRx's claims. The forward-looking statements in the press release involve risks and uncertainties, and actual results may differ materially from those projected.

In other recent news, InflaRx N.V. has been making significant strides in the development of their investigational drug, vilobelimab. The drug, also known as GOHIBIC, has been selected by the Biomedical Advanced Research and Development Authority (BARDA) for a Phase 2 clinical study. The study aims to explore new treatments for acute respiratory distress syndrome (ARDS), a critical care condition with no approved therapy.

Furthermore, InflaRx revealed promising data from a post-hoc subgroup analysis of the PANAMO Phase III study. The data suggests that vilobelimab, in combination with standard care medications, may significantly decrease mortality rates in critically ill COVID-19 patients. The study involved 369 patients and supported the emergency use authorization granted by the U.S. Food and Drug Administration (FDA) for vilobelimab in treating critically ill COVID-19 patients.

These recent developments underscore the potential of vilobelimab in the treatment of severe COVID-19 cases, although it remains investigational and has not received full FDA approval. The safety profile of vilobelimab was also assessed during the study, with no new safety concerns associated with its use in combination with other medications.

InvestingPro Insights

In light of InflaRx N.V.'s (NASDAQ:IFRX) recent presentation of preclinical data, it is important for investors to consider the company's financial health and market performance. According to InvestingPro data, InflaRx has a market capitalization of 93.62 million USD, indicating its size within the biopharmaceutical sector. The company's stock price has experienced significant volatility, with a 1-year total return of -61.69%, reflecting the high-risk nature often associated with clinical-stage biopharmaceutical companies.

InvestingPro Tips reveal that InflaRx holds more cash than debt on its balance sheet, which could provide some financial flexibility as it continues to develop its drug candidates, such as INF904. However, analysts are cautious, with two having revised their earnings estimates downwards for the upcoming period, and they do not anticipate the company will be profitable this year. This is further supported by the company's negative gross profit margin of -943.71% over the last twelve months as of Q2 2024, underscoring the challenges InflaRx faces in reaching profitability.

For investors seeking more comprehensive analysis, there are additional InvestingPro Tips available on the platform, which can provide deeper insights into InflaRx's financials, market performance, and future prospects. These tips are part of the extensive research available on InvestingPro, which includes a fair value estimate of 1.56 USD, providing a data-driven perspective on the company's valuation.

The combination of InflaRx's scientific advancements and the detailed financial data provided by InvestingPro can help investors make more informed decisions regarding their interest in the company's stock. For further detailed analysis and more InvestingPro Tips, investors can visit https://www.investing.com/pro/IFRX.

This article was generated with the support of AI and reviewed by an editor. For more information see our T&C.

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