Avacta’s pre|CISION platform shows promise in preclinical studies

Published 28/04/2025, 07:04
Avacta’s pre|CISION platform shows promise in preclinical studies

LONDON and PHILADELPHIA - Avacta Therapeutics (AIM:AVCT), a developer of peptide drug conjugates, has presented promising preclinical data for its pre|CISION® platform candidates at the American Association for Cancer Research (AACR) Annual Meeting. The event took place in Chicago, IL, where the company showcased its second pre|CISION® candidate, FAP-EXd (AVA6103), which targets the tumor microenvironment with a focus on minimizing systemic toxicity.

The pre|CISION® platform is designed to harness fibroblast activation protein-alpha (FAPα), a protease overexpressed in many solid tumors, as a means to activate anti-tumor drugs directly at the tumor site. This targeted approach aims to increase efficacy while reducing the side effects typically associated with chemotherapy.

Michelle Morrow, CSO of Avacta Therapeutics, emphasized the platform’s potential for delivering potent drugs with tumor selectivity and a novel sustained release mechanism. Morrow’s comments came as the company revealed that AVA6103, a pre|CISION® peptide drug conjugate, has shown significant tumor growth inhibition and durable complete responses in therapy-resistant preclinical models.

The compound utilizes the topoisomerase I inhibitor exatecan, which, when activated at the tumor site, displays a prolonged exposure time and the capacity to affect surrounding FAP-negative cancer cells through its bystander effect. The investigational new drug (IND) submission for FAP-EXd is expected in December 2025, with a first-in-human study slated for early 2026.

In addition to AVA6103, Avacta’s collaboration with Tempus has yielded insights into the consistent expression of FAP across different lines of therapy and tumor samples, further supporting the broad application of the pre|CISION® platform.

This news is based on a press release statement from Avacta Therapeutics and was presented at the AACR Annual Meeting. The company’s developments are being closely watched as they move towards clinical trials, which could potentially introduce new treatments for patients with solid tumors.

This article was generated with the support of AI and reviewed by an editor. For more information see our T&C.

Latest comments

Risk Disclosure: Trading in financial instruments and/or cryptocurrencies involves high risks including the risk of losing some, or all, of your investment amount, and may not be suitable for all investors. Prices of cryptocurrencies are extremely volatile and may be affected by external factors such as financial, regulatory or political events. Trading on margin increases the financial risks.
Before deciding to trade in financial instrument or cryptocurrencies you should be fully informed of the risks and costs associated with trading the financial markets, carefully consider your investment objectives, level of experience, and risk appetite, and seek professional advice where needed.
Fusion Media would like to remind you that the data contained in this website is not necessarily real-time nor accurate. The data and prices on the website are not necessarily provided by any market or exchange, but may be provided by market makers, and so prices may not be accurate and may differ from the actual price at any given market, meaning prices are indicative and not appropriate for trading purposes. Fusion Media and any provider of the data contained in this website will not accept liability for any loss or damage as a result of your trading, or your reliance on the information contained within this website.
It is prohibited to use, store, reproduce, display, modify, transmit or distribute the data contained in this website without the explicit prior written permission of Fusion Media and/or the data provider. All intellectual property rights are reserved by the providers and/or the exchange providing the data contained in this website.
Fusion Media may be compensated by the advertisers that appear on the website, based on your interaction with the advertisements or advertisers
© 2007-2025 - Fusion Media Limited. All Rights Reserved.